| 货号:23500-1 mg | 规格:1 mg | 目录价:¥482.4 |
| 货号:23500-10 mg | 规格:10 mg | 目录价:¥2492.4 |
| 货号:23500-25 mg | 规格:25 mg | 目录价:¥5065.2 |
| 货号:23500-5 mg | 规格:5 mg | 目录价:¥1809 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
CPI-637
产品描述:
An inhibitor of CBP/EP300 bromodomains (IC50s = 30 and 51 nM in a TR-FRET assay); selective for CBP and EP300 over the BET family of bromodomains (IC50s = >10 μM); is active at bromodomain BRD9 (IC50 = 0.73 μM); inhibits CBP (IC50 = 0.3 μM in a BRET assay) and inhibits MYC expression (EC50 = 0.6 μM) in AMO-1 cells
保存温度:
-20
运输温度:
-20
预期分子量:
386.5
产品形式:
A crystalline solid
有效期:
1460
纯度:
≥98%
CAS号:
1884712-47-3
分子式:
C22H22N6O
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