深圳欣博盛生物科技有限公司 a1

EHop-016
货号:21557-10 mg 规格:10 mg 目录价:¥1286
货号:21557-25 mg 规格:25 mg 目录价:¥2801
货号:21557-5 mg 规格:5 mg 目录价:¥724
货号:21557-50 mg 规格:50 mg 目录价:¥5253
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
EHop-016
产品描述:
A Rac1 and Rac3 inhibitor; inhibits Rac1 activity (IC50 = 1.1 μM); inhibits Rac3 activity (58% at 1 μM); inhibits Cdc42 activity (28% at ≥ 5 μM); increases RhoA activity (1.3-fold at ≥2 μM); increases Rac-regulated lamellipodia formation and PAK1-mediated cell migration in MDA-MB-435 cells (2-4 μM); lowers mammary fat pad tumor growth, metastasis, and angiogenesis in a nude mouse model of breast cancer (25 mg/kg); inhibits mutant KIT-induced growth in systemic mastocytosis and AML cells (≥2.5 μM)
保存温度:
-20
运输温度:
-20
预期分子量:
430.6
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
1380432-32-5
分子式:
C25H30N6O
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