深圳欣博盛生物科技有限公司 a1

ETP-46321
货号:37330-1 mg 规格:1 mg 目录价:¥700
货号:37330-10 mg 规格:10 mg 目录价:¥5600
货号:37330-25 mg 规格:25 mg 目录价:¥9632
货号:37330-5 mg 规格:5 mg 目录价:¥3164
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
ETP-46321
产品描述:
A PI3K p110α and p110δ inhibitor (apparent Kis = 2.3 and 14.2 nM, respectively); selective for PI3K p110α and p110δ over p110β and p110γ (apparent Kis = 170 and 179 nM, respectively), as well as a panel of 288 kinases at 1 µM; inhibits Akt phosphorylation in U2OS cells (IC50 = 8.3 nM); reduces tumor volume in a K-RasG12V-driven murine lung tumor model at 50 mg/kg; reduces anti-collagen IgG1 and IgG2a production, swelling, and joint rigidity in a mouse model of collagen-induced arthritis
保存温度:
-20
运输温度:
-20
预期分子量:
473.55324
产品形式:
A solid
有效期:
1460
纯度:
≥98%
CAS号:
1252594-99-2
分子式:
C20H27N9O3S
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