| 货号:45588-1 mg | 规格:1 mg | 目录价:¥656.6 |
| 货号:45588-10 mg | 规格:10 mg | 目录价:¥4931.2 |
| 货号:45588-5 mg | 规格:5 mg | 目录价:¥2787.2 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
HC-5404
别名:
LY-4
产品描述:
A PERK inhibitor (IC50 = 4 nM in a cell-free assay); selective for PERK over a panel of 25 kinases at 1 mM; reduces the levels of phosphorylated eIF2α in HEK293 cells (IC50 = 33 nM); reduces tumor volume in a 786-O mouse xenograft model at 30 mg/kg once or twice a day; has an additive effect on tumor growth inhibition when administered in combination with axitinib, cabozantinib, lenvatinib, or sunitinib in a 786-O mouse xenograft model
保存温度:
-20
运输温度:
-20
预期分子量:
454.477806
产品形式:
A solid
纯度:
≥98%
CAS号:
2247396-91-2
分子式:
C24H24F2N4O3
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