| 货号:40827-10 mg | 规格:10 mg | 目录价:¥2720 |
| 货号:40827-100 mg | 规格:100 mg | 目录价:¥20020 |
| 货号:40827-5 mg | 规格:5 mg | 目录价:¥1434 |
| 货号:40827-50 mg | 规格:50 mg | 目录价:¥11444 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
ICA 27243
别名:
ICA027243
产品描述:
An activator of Kv7.2/Kv7.3 subunit-containing channels; enhances rubidium efflux in an agonist-induced rubidium efflux assay using CHO cells expressing Kv7.2/Kv7.3 (EC50 = 0.38 µM); selective for Kv7.2/Kv7.3 channels over Kv7.4 channels (EC50 = 7.1 µM); 100-300-fold selective for Kv7.2/Kv7.3 over Kv7.3/Kv7.5 channels; selective for Kv7.2/Kv7.3 channels over a panel of neurotransmitter receptors and Nav1.2 at 10 µM, as well as GABAA receptors and high voltage-activated calcium channels at 30 µM; protects against maximal electroshock-induced seizures in a rat model of epilepsy (ED50 = 1.5 mg/kg); prevents amphetamine- and chlordiazepoxide-induced hyperactivity without affecting basal locomotor activity in a mouse model of manic-like hyperactivity at 10 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
268.7
产品形式:
A solid
纯度:
≥98%
CAS号:
325457-89-4
分子式:
C12H7ClF2N2O
促销活动
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官网链接
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