深圳欣博盛生物科技有限公司 a1

TCS 21311
货号:30063-1 mg 规格:1 mg 目录价:¥844
货号:30063-10 mg 规格:10 mg 目录价:¥4462
货号:30063-25 mg 规格:25 mg 目录价:¥10090
货号:30063-5 mg 规格:5 mg 目录价:¥2854
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
TCS 21311
别名:
NIBR3049
产品描述:
A JAK3 inhibitor (IC50 = 8 nM); selective for JAK3 over JAK1, JAK2, and TYK2 (IC50s = 1,017, 2,550, and 8,055 nM, respectively) but does inhibit GSK-3β, PKCα, and PKCθ (IC50s = 13, 68, and 3 nM, respectively); inhibits cytokine-induced STAT5 phosphorylation in CTLL and M-07 cells (IC50s = 1,294 and 525 nM, respectively) and TCR/CD28-mediated T cell activation in Jurkat cells (IC50 = 689 nM); increases proliferation of mouse embryonic NPCs and human iPSC-derived NPCs in the absence of BMP7 at 0.3 µM
保存温度:
-20
运输温度:
-20
预期分子量:
526.507169
产品形式:
A solid
纯度:
≥95%
CAS号:
1260181-14-3
分子式:
C27H25F3N4O4
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