| 货号:36938-1 mg | 规格:1 mg | 目录价:¥2706.8 |
| 货号:36938-500 µg | 规格:500 µg | 目录价:¥1420.4 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
VTX-27
产品描述:
A PKCθ inhibitor (Ki = 0.08 nM); selective for PKCθ over PKCα, -βI, -βII, -γ, -δ, -ε, -η, -µ, and -ζ (Kis = 1->5,000 nM) as well as a panel of seven kinases from the Src, Syk, Tec, and MAP kinase families (Kis = >1,000 nM for all); inhibits CD28-induced IL-2 release in isolated human PBMCs (IC50 = 11 nM); prevents staphylococcal enterotoxin B-induced increases in IL-2 plasma levels in mice at 12.5, 25, and 50 mg/kg, p.o.
保存温度:
-20
运输温度:
-20
预期分子量:
418.895503
产品形式:
A solid
有效期:
1460
纯度:
≥95%
CAS号:
1321924-70-2
分子式:
C20H24ClFN6O
促销活动
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