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折扣/货期| 货号：SIH-642-50MG | 规格：50 mg | 目录价：￥4320 |
产品详情
* 以下信息仅供参考，详情请以原厂网站为准
产品名称:
Xanomeline Tartrate
别名:
3-[4-(Hexyloxy)-1,2,5-thiadiazol-3-yl]-1,2,5,6-tetrahydro-1-methylpyridine, tartrate, LY-246708; NNC-11-0232
产品描述:
Selective muscarinic receptor agonist
保存温度:
-20ºC
运输温度:
Shipped Ambient
预期分子量:
431.5
产品形式:
Off-white powder
产地:
加拿大
生产商:
Stressmarq
功能与背景:
A functionally selective M1 muscarinic receptor agonist with high affinity for central muscarinic subtypes (EC₅₀ = 0.3, 92.5, 5, 52, and 42 nM for M1, M2, M3, M4, and M5, respectively). Its strong selectivity for M1 receptors underlies a range of central nervous system effects, including positive cognitive and behavioral improvements in models of schizophrenia and Alzheimer’s disease.
Beyond its neurocognitive actions, the compound also suppresses pro‑inflammatory cytokine responses and enhances survival in sepsis models. Additionally, it demonstrates potent analgesic efficacy in rodent models of chronic inflammatory and neuropathic pain, indicating broad therapeutic potential across neuroimmune and pain‑processing pathways.
纯度:
>98% (HPLC); NMR (Conforms)
来源:
Synthetic
CAS号:
152854-19-8
分子式:
C14H23N3OS • C4H6O6
溶解度:
May be dissolved in DMSO (45 mg/ml); or water (70 mg/ml)
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