| 货号:18011-10 mg | 规格:10 mg | 目录价:¥2265 |
| 货号:18011-25 mg | 规格:25 mg | 目录价:¥4770 |
| 货号:18011-5 mg | 规格:5 mg | 目录价:¥1206 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
XL147
别名:
Pilaralisib|SAR245408
产品描述:
A class I PI3K inhibitor (IC50s = 0.039, 0.036, 0.023, and 0.383 µM for p110α, -δ, -γ, and -β, respectively); selective for class I PI3Ks over Vps34, DNA-PK, and mTOR (IC50s = 6.974, 4.75, and >15 µM, respectively); inhibits proliferation of MCF-7 and PC3 cells (IC50s = 9.669 and 16.492 µM, respectively); reduces tumor growth in a BT474 breast cancer mouse xenograft model when administered alone or in combination with trastuzumab or lapatinib
保存温度:
-20
运输温度:
-20
预期分子量:
541
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
934526-89-3
分子式:
C25H25ClN6O4S
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