深圳欣博盛生物科技有限公司 a1

AZ9482
货号:SYN-3046-M001 规格:1 mg 目录价:¥1358
货号:SYN-3046-M005 规格:5 mg 目录价:¥2870
货号:SYN-3046-M010 规格:10 mg 目录价:¥4382
货号:SYN-3046-M050 规格:50 mg 目录价:¥13454
货号:SYN-3046-M100 规格:100 mg 目录价:¥询价
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
AZ9482
别名:
2-(4-(3-((4-Oxo-3,4-dihydrophthalazin-1-yl)methyl)benzoyl)piperazin-1-yl)nicotinonitrile
产品描述:
AZ9482 is a potent and selective PARP inhibitor featuring an amide linkage to a 2-piperazinyl-3-cyano-pyridine. AZ9482 exhibits very potent centrosome declustering activity in HeLa cells (EC50 < 18nM). AZ9482 also showed a 3nM GI50 in the DLBCL cell line OCI-LY-19 in a 3-day AlamarBlue assay. Consistent with published siRNA knockdown experiments, AZ9482 was a 9nM enzyme inhibitor of tankyrase 1 (TNKS1).
保存温度:
+4°C
运输温度:
Ambient
预期分子量:
450.5
产品形式:
solid
有效期:
Stable for at least 2 years after receipt when stored at -20°C.
产地:
瑞士
纯度:
>95%
CAS号:
1825345-33-2
分子式:
C26H22N6O2
溶解度:
Soluble in DMSO or ethanol.
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