深圳欣博盛生物科技有限公司 a1

Derenofylline
货号:27666-1 mg 规格:1 mg 目录价:¥509
货号:27666-10 mg 规格:10 mg 目录价:¥2452
货号:27666-25 mg 规格:25 mg 目录价:¥5481
货号:27666-5 mg 规格:5 mg 目录价:¥1367
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Derenofylline
别名:
SLV 320
产品描述:
An adenosine A1 receptor antagonist (Ki = 1 nM); selective for adenosine A1 over A2A, A2B, and A3 receptors (Kis = 398, 3,981, and 200 nM, respectively); decreases adenosine A1 receptor-mediated adenosine-induced bradycardia in rats (ED50 = 0.49 mg/kg) but reduces A2 receptor-mediated adenosine-induced hypotension by only 44.6% at an intravenous dose of 5 mg/kg; prevents increases in heart levels of collagen I and III in nephrectomized rats at 10 mg/kg per day; reduces relative plaque counts in a Zika virus plaque-forming assay in A549 cells (IC50 = 58.6 nM) in an adenosine A1 receptor-independent manner
保存温度:
-20
运输温度:
-20
预期分子量:
308.37776
产品形式:
A solid
纯度:
≥98%
CAS号:
251945-92-3
分子式:
C18H20N4O
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