深圳欣博盛生物科技有限公司 a1

Elacestrant (hydrochloride)
货号:37298-1 mg 规格:1 mg 目录价:¥1018.4
货号:37298-10 mg 规格:10 mg 目录价:¥7906
货号:37298-5 mg 规格:5 mg 目录价:¥4489
货号:37298-500 µg 规格:500 µg 目录价:¥536
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Elacestrant (hydrochloride)
别名:
RAD901
产品描述:
A selective estrogen receptor degrader; selectively binds to ERα over ERβ (IC50s = 48 and 870 nM, respectively) and reduces ERα levels in MCF-7 cells (EC50 = 0.6 nM); reduces E2-induced MCF-7 proliferation (EC50 = 4 pM); reduces E2-induced tumor growth in an MCF-7 mouse xenograft model at 30 and 60 mg/kg; increases survival in an MCF-7 intracranial mouse xenograft model; protects against bone loss in ovariectomized rats from 0.1-3 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
531.6
产品形式:
A solid
有效期:
1460
纯度:
≥98%
CAS号:
1349723-93-8
分子式:
C30H38N2O2 • 2HCl
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