| 货号:SYN-1221-M001 | 规格:1 mg | 目录价:¥1204 |
| 货号:SYN-1221-M005 | 规格:5 mg | 目录价:¥2870 |
| 货号:SYN-1221-M010 | 规格:10 mg | 目录价:¥4382 |
| 货号:SYN-1221-M050 | 规格:50 mg | 目录价:¥询价 |
| 货号:SYN-1221-M100 | 规格:100 mg | 目录价:¥询价 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
H-1152
别名:
(S)-4-Methyl-5-((2-methyl-1,4-diazepan-1-yl)sulfonyl)isoquinoline dihydrochloride; H1152
产品描述:
H-1152 is a potent, specific, ATP-competitive and cell permeable ROCK inhibitor, with an IC50 of 12nM for ROCKII. H-1152 poorly inhibits PKA, PKC and myosin light chain kinase. Rho kinase (ROCK) activated by GTP-linked Rho phosphorylates targets that are involved in cytoskeletal remodelling, smooth muscle contraction and neuronal development.
保存温度:
+4°C
运输温度:
Ambient
预期分子量:
319.4 . 72.9
产品形式:
solid
产地:
瑞士
纯度:
>95%
CAS号:
871543-07-6
分子式:
C16H21N3O2S . 2HCl
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