深圳欣博盛生物科技有限公司 a1

Momelotinib
货号:SYN-1035-M001 规格:1 mg 目录价:¥1204
货号:SYN-1035-M005 规格:5 mg 目录价:¥1666
货号:SYN-1035-M010 规格:10 mg 目录价:¥2422
货号:SYN-1035-M050 规格:50 mg 目录价:¥6804
货号:SYN-1035-M100 规格:100 mg 目录价:¥询价
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Momelotinib
别名:
CYT387; Momelotinib
产品描述:
CYT387 is selective inhibitor of JAK1 and JAK2 kinases including the JAK2V617F mutant . Using ATP kinase assays IC(50) values for JAK1 (11nm), JAK2, (18nM), JAK2, JAK2V617F (23nM) JAK3 (155nM), and TYK2 (17nM). In testing kinase arrays, CYT387 also had activity (defined as an IC(50) < 100nM) detected against CDK2/cyclin A, MAPK8 (JNK1), PRKCN (PKD3), PRKD1 (PKCµ), ROCK2, and TBK1 kinase as well.
保存温度:
+4°C
运输温度:
Ambient
预期分子量:
414.5
产品形式:
solid
有效期:
Stable for at least 2 years after receipt when stored at -20°C.
产地:
瑞士
纯度:
>95%
CAS号:
1056634-68-4
分子式:
C23H22N6O2
溶解度:
Soluble in DMSO.
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