| 货号:SYN-1035-M001 | 规格:1 mg | 目录价:¥1204 |
| 货号:SYN-1035-M005 | 规格:5 mg | 目录价:¥1666 |
| 货号:SYN-1035-M010 | 规格:10 mg | 目录价:¥2422 |
| 货号:SYN-1035-M050 | 规格:50 mg | 目录价:¥6804 |
| 货号:SYN-1035-M100 | 规格:100 mg | 目录价:¥询价 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Momelotinib
别名:
CYT387; Momelotinib
产品描述:
CYT387 is selective inhibitor of JAK1 and JAK2 kinases including the JAK2V617F mutant . Using ATP kinase assays IC(50) values for JAK1 (11nm), JAK2, (18nM), JAK2, JAK2V617F (23nM) JAK3 (155nM), and TYK2 (17nM). In testing kinase arrays, CYT387 also had activity (defined as an IC(50) < 100nM) detected against CDK2/cyclin A, MAPK8 (JNK1), PRKCN (PKD3), PRKD1 (PKCµ), ROCK2, and TBK1 kinase as well.
保存温度:
+4°C
运输温度:
Ambient
预期分子量:
414.5
产品形式:
solid
产地:
瑞士
纯度:
>95%
CAS号:
1056634-68-4
分子式:
C23H22N6O2
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