| 货号:SYN-1194-M001 | 规格:1 mg | 目录价:¥2954 |
| 货号:SYN-1194-M005 | 规格:5 mg | 目录价:¥5824 |
| 货号:SYN-1194-M010 | 规格:10 mg | 目录价:¥9142 |
| 货号:SYN-1194-M050 | 规格:50 mg | 目录价:¥询价 |
| 货号:SYN-1194-M100 | 规格:100 mg | 目录价:¥询价 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
PF-04979064
别名:
PF04979064
产品描述:
PF-04979064 is a potent and selective PI3K/mTOR dual kinase inhibitor with an IC(50) of 9.1nM for the PI3K family when tested AKT phosphorylation in BT20 cells. In direct kinase assays, PF-04979064 has potent Ki values against PI3Kalpha (Ki= 0.13nM human, 0.299nM mouse) and PI3Kgamma (Ki=0.111nM), and PI3Kdelta (Ki=0.122nM). In contrast, Ki values for non-PI3K kinases such as mTOR were 10X higher at 1.42 nM.
保存温度:
+4°C
运输温度:
Ambient
预期分子量:
446.5
产品形式:
solid
产地:
瑞士
纯度:
>95%
CAS号:
1220699-06-8
分子式:
C24H26N6O3
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