| 货号:AG-CR1-3647-M001 | 规格:1 mg | 目录价:¥1440 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Jak/Src Inhibitor 1 . hydrochloride
别名:
Debio 0617B . HCl; N-(4-Chloro-3-(2-((4-(methyl-carbamoyl)phenyl)amino)-7,8-dihydropyrido[4,3-d]pyrimidin-6(5H)-yl)phenyl)-4-(trifluoromethyl)picolinamide
产品描述:
Multi-kinase inhibitor with potent antiproliferative anti-migratory activities. Potent STAT3/5 inhibitor in vitro and in vivo. Combined inhibitor of key kinases phosphorylating STAT3 and STAT5 proteins such as JAK, SRC, ABL families of kinases, and class III/V receptor tyrosine kinases (RTK), including FLT3, c-KIT, CSF1-R, PDGFRs and VEGFRs, in nanomolar range.
保存温度:
+4°C
运输温度:
Ambient
预期分子量:
582.0 . 36.5
产品形式:
solid
产地:
瑞士
纯度:
>97% (HPLC)
CAS号:
1332329-27-7 (parent)
分子式:
C28H23ClF3N7O2 . HCl
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